Pasireotide (diaspartate)

SKU: orb1982174

Description

Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, <7.0, and 9.9, respectively). This compound demonstrates antisecretory, antiproliferative, and proapoptotic activities.

Images & Validation

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Key Properties

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CAS Number	1421446-02-7
MW	1313.41
Formula	C₆₆H₈₀N₁₂O₁₇
SMILES	OC(C[C@H](N)C(O)=O)=O.O=C1N2[C@@](C(N[C@@H](C3=CC=CC=C3)C(N[C@@H](C(N[C@H](C(N[C@H](C(N[C@H]1CC4=CC=CC=C4)=O)CC5=CC=C(C=C5)OCC6=CC=CC=C6)=O)CCCCN)=O)CC7=CNC8=CC=CC=C78)=O)=O)([H])C[C@H](C2)OC(NCCN)=O.OC(C[C@H](N)C(O)=O)=O
Target	Others,Somatostatin

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Gene Symbol

Others,Somatostatin

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