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Avapritinib

SKU: orb1225956

Description

Avapritinib (BLU-285) is a potent and highly selective inhibitor of mutant KIT and PDGFRα with IC50 of 0.6, 0.27 and 0.24 nM for KIT del557-558, KIT D816V and PDGFRA D842V, respectively.

Images & Validation

Key Properties

CAS Number1703793-34-3
MW498.6
Purity>98% (HPLC)
FormulaC26H27FN10
TargetKITD816V|PDGFRαD842V

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
DisclaimerFor research use only

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    200 mg, 25 mg, 10 mg, 5 mg, 100 mg, 50 mg, 1 mg, 1 ml x 10 mM (in DMSO)
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Avapritinib (orb1225956)

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Available Sizes

Select a size below

5 mg
$ 290.00
10 mg
$ 450.00
25 mg
$ 710.00
50 mg
$ 1,010.00
100 mg
$ 1,330.00
500 mg
$ 2,640.00