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Sepimostat

SKU: orb1298524

Description

Sepimostat dimethanesulfonate is a neuroprotective agent that functions as an NR2B NMDA receptor antagonist, competitively inhibiting ifenprodil binding with a Ki of 27.7 µM. This activity supports its research use in studying excitotoxicity and neuronal injury in both cellular and animal models of stroke and neurodegenerative diseases.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number103926-64-3
MW373.41
Purity99.30% (May vary between batches)
FormulaC21H19N5O2
SMILESNC(=N)c1ccc2cc(OC(=O)c3ccc(NC4=NCCN4)cc3)ccc2c1
TargetiGluR
SolubilityDMSO:6.25 mg/mL (16.74 mM)

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

Ionotropic glutamate receptors, NR2B N-methyl-D-aspartate, inhibit, iGluR, Inhibitor, FUT 187, FUT187, FUT-187, Sepimostat

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Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

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Sepimostat (orb1298524)

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% DMSO +
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% Tween 80 +
%

Available Sizes

Select a size below

1 mg
$ 90.00
5 mg
$ 160.00
1 ml x 10 mM (in DMSO)
$ 170.00
10 mg
$ 240.00
25 mg
$ 380.00
50 mg
$ 520.00
100 mg
$ 700.00
200 mg
$ 930.00
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