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β2AR/M-receptor agonist-1

SKU: orb1982697

Description

β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and muscarinic receptor, with an EC50 value of 9.2 nM for β2 adrenoceptor and a Ki value of 30.2 nM for the muscarinic receptor, and an EC50 value of 4.0 nM highlighting its MABA activity.

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Key Properties

CAS Number2230520-62-2
MW806.82
FormulaC43H56BrN3O7
SMILES[Br-].O[C@H](CNCCCOc1ccc(OCCC[N+]23CCC(CC2)[C@@H](C3)OC[C@@](O)(C2CCCC2)c2ccccc2)cc1)c1ccc(O)c2[nH]c(=O)ccc12
TargetAChR,Others,Adrenergic Receptor

Storage & Handling

Storage-20°C
DisclaimerFor research use only
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β2AR/M-receptor agonist-1 (orb1982697)

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