β2AR/M-receptor agonist-2

SKU: orb1745044

Description

β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA). It demonstrates significant activity towards the β2 adrenoceptor with an EC50 of 3.7 nM and exhibits affinity for the human cloned M3 receptor with a Ki of 0.73 nM. This potent bronchodilator holds potential for research in chronic obstructive pulmonary disease (COPD) treatment.

Images & Validation

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Key Properties

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CAS Number	1017857-38-3
MW	717.31
Formula	C₃₆H₄₉ClN₄O₇S
SMILES	N(C(OC1CCN(CCCCCCCCCNC[C@H](O)C2=CC(NS(C)(=O)=O)=C(O)C=C2)CC1)=O)C3=C(C=CC=C3)C4=CC(Cl)=C(O)C=C4
Target	AChR,Others,Adrenergic Receptor

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Gene Symbol

AChR,Others,Adrenergic Receptor

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