5-HT2A/5-HT2C inverse agonist 1

SKU: orb2665522

Description

5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A and 5-HT2C receptors, with hERG inhibition properties that mitigate cardiovascular risks. Demonstrating significant antipsychotic efficacy in the MK-801-induced mouse model, this compound holds potential for psychosis research.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	2718990-76-0
MW	425.57
Formula	C₂₄H₃₅N₅O₂
SMILES	N(CC1=NN(C)C=C1)(C(NCC2=CC=C(OCCC)C=C2)=O)[C@@H]3C4(CC4)CN(C)CC3
Target	5-HT Receptor

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Gene Symbol

5-HT Receptor

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