[Ala17]-MCH acetate

SKU: orb1296398

Description

[Ala17]-MCH acetate is a potent and selective MCHR1 antagonist, exhibiting high affinity (Ki = 0.16 nM) and over 200-fold selectivity versus MCHR2. This tool compound is valuable for investigating the role of the MCH system in energy homeostasis, sleep, and mood regulation in both in vitro binding assays and in vivo preclinical models.

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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Target	Melanin-concentrating Hormone Receptor (MCHR)
Molecular Weight	2331.76
Purity	98.92%
Formula	C₉₉H₁₅₉N₂₉O₂₈S₄
SMILES	O=C1N2[C@](CCC2)([H])C(N[C@@H](CSSC[C@@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]1CCCNC(N)=N)=O)CC3=CC=C(C=C3)O)=O)C(C)C)=O)CCCNC(N)=N)=O)=O)CC(C)C)=O)CCSC)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@H](CCSC)NC([C@H](CC(O)=O)NC([C@@H](NC([C@@H](N)CC(O)=O)=O)CC4=CC=CC=C4)=O)=O)=O)=O)=O)C(N[C@@H](C)C(N[C@@H](CCC(N)=O)C(N[C@H](C(O)=O)C(C)C)=O)=O)=O)=O.CC(O)=O

Storage & Handling

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Storage	store at low temperature,keep away from moisture \| Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Alternative Names

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[Ala17]-MCH Acetate, [Ala17]-MCH acetate(359784-84-2 free base), Melanin-concentrating Hormone Receptor, Melaninconcentrating Hormone Receptor (MCHR), MelaninconcentratingHormoneReceptor, MelaninconcentratingHormoneReceptor(MCHR), MCH1-R, MCHR, MCHR2

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Compound Identifiers

PubChem CID

176418218 ↗

Key Properties

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No computed properties available.

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