Desmethylazelastine

SKU: orb1982811

Description

Desmethylazelastine, the primary active metabolite of Azelastine, undergoes oxidative metabolism via the cytochrome P450 enzyme system, exhibits a 97% protein binding rate, and has an elimination half-life of 54 hours. Azelastine, an orally active, selective, and high-affinity histamine H1-receptor antagonist, is utilized in the research of allergic rhinitis, asthma, diabetic hyperlipidemia, and SARS-CoV-2.

Research Area

Metabolism Research

Images & Validation

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Key Properties

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CAS Number	47491-38-3
MW	367.87
Formula	C₂₁H₂₂ClN₃O
SMILES	Clc1ccc(Cc2nn(C3CCCNCC3)c(=O)c3ccccc23)cc1
Target	Drug Metabolite,Others

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Gene Symbol

Drug Metabolite,Others

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