Firazorexton hydrate

SKU: orb2278508

Description

Firazorexton hydrate (TAK-994) is a brain-penetrant, orally active agonist of the orexin type 2 receptor (OX2R) with a potent EC50 of 19 nM, effectively reducing wakefulness fragmentation and cataplexy-like episodes in mouse models of narcolepsy.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	2861934-86-1
MW	497.53
Formula	C₂₂H₂₅F₃N₂O₄S.3/2H₂O
SMILES	C([C@@H]1N(C(C(C)(C)O)=O)CC[C@@H]1NS(C)(=O)=O)C2=C(F)C(=CC=C2)C3=CC(F)=CC(F)=C3.O
Target	OX Receptor,Others

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Gene Symbol

OX Receptor,Others

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