Cart summary

You have no items in your shopping cart.

G-1

SKU: orb1308286

Description

G-1 is a nonsteroidal, high-affinity, and selective agonist for GPR30 (GPER), with a Ki value of 11 nM. This compound is employed in both in vitro and in vivo research to study GPER-mediated signaling in fields such as oncology, cardiology, endocrinology, and neuroscience, as documented in scientific literature.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number881639-98-1
MW412.28
Purity99.89%
FormulaC21H18BrNO3
SMILES[H][C@@]12CC=C[C@]1([H])c1cc(ccc1N[C@@H]2c1cc2OCOc2cc1Br)C(C)=O
TargetGPCR,Estrogen Receptor/ERR
SolubilityDMSO:120 mg/mL (291.06 mM);H2O:< 0.1 mg/mL (insoluble);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.85 mM)

Storage & Handling

Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
DisclaimerFor research use only

Alternative Names

ERR, G 1, Estrogen Receptor/ERR, EstrogenReceptor, Estrogen Receptor, GPR30, G1, G-1, inhibit, Inhibitor

Similar Products

  • ANXA5 Antibody [orb242618]

    ELISA,  IHC,  WB

    Human

    Rabbit

    Polyclonal

    Unconjugated

    100 μg, 50 μg
  • Human Pregnancy Specific Beta-1-Glycoprotein 1 (PSG1/SP1) ELISA Kit [orb1948570]

    Human

    3.13-200ng/mL

    1.88 ng/mL

    48 T, 96 T
  • PSG1 rabbit pAb Antibody [orb766858]

    ELISA,  IF,  IHC,  WB

    Human, Mouse, Rat

    Polyclonal

    Unconjugated

    50 μl, 100 μl
  • Celery (api g 1) [orb1925098]

    CLIA,  ELISA,  LF,  WB

    100 μg
  • rApi g 1 (Apium graveolens 1.0101) Antibody [orb1088535]

    ELISA,  FC

    Unconjugated

    0.1 mg
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at support@biorbyt.com.

Documents Download

Datasheet
Product Information
Download

Request a Document

Protocol Information

G-1 (orb1308286)

  • Star
  • Star
  • Star
  • Star
  • Star
  • 0.0
Based on 0 reviews

Participating in our Biorbyt product reviews program enables you to support fellow scientists by sharing your firsthand experience with our products.

Login to Submit a Review

No reviews yet

Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

(This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

1 mg
$ 90.00
1 ml x 10 mM (in DMSO)
$ 120.00
5 mg
$ 120.00
10 mg
$ 170.00
25 mg
$ 260.00
50 mg
$ 380.00
100 mg
$ 530.00
200 mg
$ 740.00
DispatchUsually dispatched within 3-5 working days
Bulk Enquiry