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H3R antagonist 5

SKU: orb2944544

Description

H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.

Research Area

Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number879368-27-1
MW400.511
FormulaC23H32N2O4
SMILESO=C1O[C@]2(C=3C1=CC(OC)=CC3)CC[C@@H](C(N(CCN4CCCCC4)C)=O)CC2
TargetHistamine Receptor

Storage & Handling

Storage-20°C
DisclaimerFor research use only
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H3R antagonist 5 (orb2944544)

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