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LAS190792

SKU: orb1982696

Description

LAS190792 (AZD8999) is a dual-action chemical compound that simultaneously acts as a strong muscarinic antagonist and β2-adrenoceptor agonist. It exhibits significant potency across a range of receptors, with pIC50 values of 8.9 for M1, 8.8 for M2, 8.8 for M3, 9.2 for M4, 8.2 for M5, 7.5 for β1, 9.1 for β2, and 5.6 for β3. Its effectiveness across these receptors makes LAS190792 a viable candidate for bronchodilator applications.

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Key Properties

CAS Number1347232-69-2
MW811.36
FormulaC39H43ClN4O9S2
SMILESCOc1cc(NC(=O)OCCN(C)[C@H]2CC[C@@H](CC2)OC(=O)C(O)(c2cccs2)c2cccs2)c(Cl)cc1CNC[C@H](O)c1ccc(O)c2[nH]c(=O)ccc12
TargetOthers,Adrenergic Receptor,AChR

Storage & Handling

Storage-20°C
DisclaimerFor research use only
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LAS190792 (orb1982696)

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