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TGR5 Receptor Agonist 4

SKU: orb1943763

Description

TGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5). It is notably involved in mediating hypoglycemic and weight loss effects.

Images & Validation

Key Properties

CAS Number1872436-42-4
MW470.95
FormulaC25H27ClN2O5
SMILESC(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4
TargetOthers

Storage & Handling

Storage-20°C
DisclaimerFor research use only

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TGR5 Receptor Agonist 4 (orb1943763)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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